Synthesis and Preclinical Evaluation of Urea-Based Prostate-Specific Membrane Antigen-Targeted Conjugates Labeled with 177Lu

Авторы
Machulkin Aleksei E. 2, 1 , Petrov Stanislav A. 1 , Bodenko Vitalina 3, 4 , Larkina Mariia S. 3, 5 , Plotnikov Evgenii 6, 3 , Yuldasheva Feruza 3 , Tretyakova Maria 3 , Bezverkhniaia Ekaterina 3, 7 , Zyk Nikolay Yu. 1 , Stasyuk Elena 8 , Zelchan Roman 3 , Majouga Alexander G. 9 , Tolmachev Vladimir 10 , Orlova Anna 7 , Beloglazkina Elena K. 1 , Yusubov Mekhman S. 3
Издательство
American Chemical Society
Номер выпуска
5
Язык
Английский
Страницы
1457-1473
Статус
Опубликовано
Том
7
Год
2024
Организации
  • 1 Department of Chemistry, M.V. Lomonosov Moscow State University, Leninskie Gory 1-3, Moscow 119991, Russian Federation
  • 2 Department for Biochemistry, People’s Friendship University of Russia Named after Patrice Lumumba (RUDN University), Moscow 117198, Russia
  • 3 Research Centrum for Oncotheranostics, Research School of Chemistry and Applied Biomedical Sciences, Tomsk Polytechnic University, Tomsk 634050, Russia
  • 4 Scientific and Educational Laboratory of Chemical and Pharmaceutical Research, Siberian State Medical University, Tomsk 634050, Russia
  • 5 Department of Pharmaceutical Analysis, Siberian State Medical University, Tomsk 634050, Russia
  • 6 Mental Health Research Institute, Tomsk National Research Medical Center, Russian Academy of Sciences, Tomsk 634014, Russia
  • 7 Department of Medicinal Chemistry, Uppsala University, Uppsala 75183, Sweden
  • 8 School of Nuclear Science and Engineering, Tomsk Polytechnic University, Tomsk 634050, Russia
  • 9 Dmitry Mendeleev University of Chemical Technology of Russia, Miusskaya sq. 9, Moscow 125047, Russian Federation
  • 10 Department of Immunology, Genetics and Pathology, Uppsala University, Uppsala 75185, Sweden
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