DESIGN OF NEW ANTI-ALZHEIMER DRUGS: RING-EXPANSION SYNTHESIS AND SYNCHROTRON X-RAY DIFFRACTION STUDY OF DIMETHYL 4-ETHYL-11-FLUORO-1,4,5,6,7,8-HEXAHYDROAZONINO[5,6-B]INDOLE-2,3-DICARBOXYLATE ArticleToze F.A.A., Listratova A.V., Voskressensky L.G., Chernikova N.Yu., Lobanov N.N., Bilyachenko A.N., Dorovatovskii P.V.Acta Crystallographica Section E: Crystallographic Communications. Том 74. 2018. С. 298-301
THREE-COMPONENT REACTION BETWEEN ISATOIC ANHYDRIDE, AMINE AND METH-YL-SUBS-TITUTED FURYL-ACRYL-ALDE-HYDES: CRYSTAL STRUCTURES OF 3-BENZYL-2-[(E)-2-(5-METHYLFURAN-2-YL)VIN-YL]-2,3-DI-HYDRO-QUINAZOLIN-4(1 H)-ONE, 3-BENZYL-2-[(E)-2-(FURAN-2-YL)-1-METHYL-VIN-YL]-2,3-DI-HYDRO-QUINAZOLIN-4(1 H)-ONE AND 3-(FURAN-2-YLMETH-YL)-2-[(E)-2-(FURAN-2-YL)-1-METHYL-VIN-YL]-2,3-DI-HYDRO-QUINAZOLIN-4(1 H)-ONE ArticleZaytsev V.P., Sorokina E.A., Kvyatkovskaya E.A., Toze F.A.A., Mhaldar S.N., Dorovatovskii P.V., Khrustalev V.N.Acta Crystallographica Section E: Crystallographic Communications. Том 74. 2018. С. 1101-1106
CRYSTAL STRUCTURE OF 3-BENZYL-2-[(E)-2-(FURAN-2-YL)ETHENYL]-2,3-DIHYDROQUINAZOLIN-4(1H)-ONE AND 3-BENZYL-2-[(E)-2-(THIOPHEN-2-YL)ETHENYL]-2,3-DIHYDROQUINAZOLIN-4(1H)-ONE FROM SYNCHROTRON X-RAY DIFFRACTION ArticleToze F.A.A., Zaytsev V.P., Chervyakova L.V., Kvyatkovskaya E.A., Dorovatovskii P.V., Khrustalev V.N.Acta Crystallographica Section E: Crystallographic Communications. Том 74. 2018. С. 10-14
CRYSTAL STRUCTURES OF (5RS)-(Z)-4-[5-(FURAN-2-YL)-3-PHENYL-4,5-DIHYDRO-1H-PYRAZOL-1-YL]-4-OXOBUT-2-ENOIC ACID AND (5RS)-(Z)-4-[5-(FURAN-2-YL)-3-(THIOPHEN-2-YL)-4,5-DIHYDRO-1H-PYRAZOL-1-YL]-4-OXOBUT-2-ENOIC ACID ArticleBorisova K.K., Toze F.A.A., Yagafarov N.Z., Zubkov F.I., Dorovatovskii P.V., Zubavichus Y.V., Khrustalev V.N.Acta Crystallographica Section E: Crystallographic Communications. Том 72. 2016. С. 1557-1561
SYNTHESIS OF FURYL-, FURYLVINYL-, THIENYL-, PYRROLINYLQUINAZOLINES AND ISOINDOLO[2,1-A]QUINAZOLINES ArticleZaytsev V.P., Revutskaya E.L., Kuźmenko M.G., Novikov R.A., Zubkov F.I., Sorokina E.A., Nikitina E.V., Toze F.A.A., Varlamov A.V.Russian Chemical Bulletin. Том 64. 2015. С. 1345-1353
SYNTHESIS OF 2-(CHLORO(METHOXY, MORPHOLINO)METHYL)-HEXAHYDROPYRIMIDOTHIENO[3,2-C]AZOCINES AND TETRAHYDROSPIRO[PYRIDO[4,5']THIENO[2,3-D]PYRIMIDINES] ArticleVoskressensky L.G., Kovaleva S.A., Borisova T.N., Titov A.A., Toze F., Listratova A.V., Khrustalev V.N., Varlamov A.V.Chemistry of Heterocyclic Compounds. Том 51. 2015. С. 17-25
CRYSTAL STRUCTURE OF METHYL (3RS,4SR,4ARS,11ARS,11BSR)-5-OXO-3,4,4A,5,7,8,9,10,11,11A-DECAHYDRO-3,11B-EPOXYAZEPINO[2,1-A]ISOINDOLE-4-CARBOXYLATE ArticleToze F.A.A., Poplevin D.S., Zubkov F.I., Nikitina E.V., Porras C., Khrustalev V.N.Acta Crystallographica Section E: Crystallographic Communications. Том 71. 2015. С. o729-o730
THE INTERACTION OF 4-HYDROXYMETHYL ISOINDOLINES WITH DEHYDROBENZENE. SYNTHESIS OF 3-PHENYLAMINOMETHYLDIHYDROBENZO[C]FURANES ArticleVarlamov A.V., Guranova N.I., Borisova T.N., Toze F.A.A., Ovcharov M.V., Kristancho S., Voskressensky L.G.Tetrahedron. Том 71. 2015. С. 1175-1181
TRANSFORMATIONS OF 4-ARYLPYRROLO[1,2-A][1,4]BENZODIAZEPINES IN THREE-COMPONENT REACTIONS WITH ACTIVATED ALKYNES AND СН, NH, SH, AND ОН ACIDS ArticleVoskressensky L.G., Borisova T.N., Babakhanova M.I., Chervyakova T.M., Titov A.A., Novikov R.A., Toze F., Dang T.T.A., Varlamov A.V.Chemistry of Heterocyclic Compounds. Том Vol 51. 2015. С. 639-646
TRANSFORMATIONS OF 4-ARYLPYRROLO[1,2-A][1,4]BENZODIAZEPINES IN THREE-COMPONENT REACTIONS WITH ACTIVATED ALKYNES AND CH, NH, SH, AND OH ACIDS ArticleVoskressensky L.G., Borisova T.N., Babakhanova M.I., Chervyakova T.M., Titov A.A., Novikov R.A., Toze F., Dang T.T.A., Varlamov A.V.Chemistry of Heterocyclic Compounds. Том 51. 2015. С. 639-646
5-AMIDO- AND 5-AMINO-SUBSTITUTED EPOXYISOINDOLO[2,1-A]TETRAHYDROQUINOLINES AND 10-CARBOXYLIC ACIDS: THEIR SYNTHESIS AND REACTIVITY ArticleZaytsev V.P., Zubkov F.I., Toze F.A.A., Orlova D.N., Eliseeva M.N., Grudinin D.G., Nikitina E.V., Varlamov A.V.Journal of Heterocyclic Chemistry. Том 50. 2013. С. E18-E38
RAC-METHYL (3AR*,4S*,5R*,7AR*)-5,7A-BIS(ACETYLOXY)- 3-OXO-2-PHENYLOCTAHYDRO-1H-ISOINDOLE-4-CARBOXYLATE ArticleToze F.A.A., Nikitina E.V., Zaytsev V.P., Zubkov F.I., Khrustalev V.N.Acta Crystallographica Section E: Structure Reports Online. Том 69. 2013. o1555 с.
METHYL (9AR*,10S*,11R*,13AS*,13BS*)-9-OXO-6, 7,9,9A,10,11-HEXAHYDRO-5H,13BH-11,13A-EPOXYPYRROLO-[2′,1′:3,4][1,4] DIAZEPINO[2,1-A]ISOINDOLE-10-CARBOXYLATE ArticleToze F.A.A., Airiyan I.K., Nikitina E.V., Sorokina E.A., Khrustalev V.N.Acta Crystallographica Section E: Structure Reports Online. Том 67. 2011. С. o2852-o2853
8A-METHYL-5,6,8,8A,9,10-HEXA-HYDRO-10,12A-EPOXY-ISOINDOLO[1,2-A] ISOQUINOLINIUM IODIDE ArticleToze F.A.A., Ershova J.D., Obushak M.D., Zubkov F.I., Khrustalev V.N.Acta Crystallographica Section E: Structure Reports Online. Том 66. 2010. С. o1388-o1389
FIRST EXAMPLE OF DIELS-ALDER REACTION IN THE 2,3,4,4A-TETRAHYDROQUINOLINE SERIES. SYNTHESIS OF HYDROGENATED 5,8-ETHANOQUINOLINES ArticleNikitina E.V., Khrustalev V.N., Grudinin D.G., Toze F.A.A., Kouznetsov V.V., Zubkov F.I.Tetrahedron. Том 66. 2010. С. 2889-2894